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derivatives designed derivatives derivative synthesis anti model molecular antitubercular activity tema motivador dihydrofolate reductase oxazolidine derivative trifluoromethyl drug plasmodium falciparum oficinas pedagogicas novo analogo mefloquine lassbio qsar acylhydrazone quimica acylhydrazone derivative qsar analysis antimalarial inibidores seletivos derivados alunos ensino inhibitor