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sintese anti meninas quimica leishmanicidal derivatives quimica evaluation inibidores seletivos oficinas pedagogicas inhibitor novel qsar analysis ensino medio derivatives designed model oxazolidine derivative lassbio analogo mefloquine dihydrofolate reductase drug pharmacological evaluation acylhydrazone derivative synthesis plasmodium falciparum activity acylhydrazone derivados antitubercular tema motivador